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METHODS Terazosin hydrochloride was synthesized from anhydro-piperazine via acylation,reduction,amination,salification etc.

方法以无水哌嗪为起始,酰化、还、胺化、成等反制得酸特拉唑嗪。

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The title resin has been prepared by Friedel-Crafts acylation followed by bromination and amination.The method avoids the utilization of cancerogenic chloromethyl methyl ether.

通过付氏酰基化反乙酰基,接着溴化、胺化,得到标题树脂。该法避免了使用氯甲醚。

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